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ChEMBL ligand: CHEMBL1521056 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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CysLT1 receptor in Human [GtoPdb: 269] [UniProtKB: Q9Y271] | ||||||||
GtoPdb | - | - | 9.3 | pKd | 0.5 | nM | Kd | Prostaglandins Other Lipid Mediat (2003) 71: 235-51 [PMID:14518564] |
GtoPdb | - | - | 10.22 | pKd | - | - | Kd |
Nature (1999) 399: 789-93 [PMID:10391245]; J Cell Sci (2005) 118: 5625-36 [PMID:16306225] |
GtoPdb | - | - | 10.6 | pKd | - | - | - |
Mol Pharmacol (1998) 53: 750-8 [PMID:9547367]; Br J Pharmacol (1998) 123: 590-8 [PMID:9504401] |
GtoPdb | - | - | 10.7 | pKd | 0.02 | nM | Kd | |
CysLT2 receptor in Human [GtoPdb: 270] [UniProtKB: Q9NS75] | ||||||||
GtoPdb | - | - | 9.4 | pKd | 0.4 | nM | Kd | J Biol Chem (2000) 275: 30531-6 [PMID:10851239] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]