(-)-bremazocine [Ligand Id: 1603] activity data from GtoPdb

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  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
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  • κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
  • κ receptor in Mouse [GtoPdb: 318] [UniProtKB: P33534]
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  • μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb - - 9 pKi - - - NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
GtoPdb - - 10.5 pKi - - - NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]
κ receptor in Mouse [GtoPdb: 318] [UniProtKB: P33534]
GtoPdb - - 9.5 pIC50 - - - Proc Natl Acad Sci USA (1993) 90: 6736-40 [PMID:8393575]
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
GtoPdb - - 9.7 pKi - - - NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.