pasireotide [Ligand Id: 2018] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | - | - | - | Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717] |
| SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | - | - | - | Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717] |
| SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680] | ||||||||
| GtoPdb | - | - | 5 | pEC50 | >10000 | nM | EC50 | Mol Endocrinol (2010) 24: 240-9 [PMID:19910453] |
| GtoPdb | - | - | 7.63 | pEC50 | 23.3 | nM | EC50 | Mol Endocrinol (2011) 25: 1040-54 [PMID:21493671] |
| GtoPdb | - | - | 9.07 | pEC50 | 0.86 | nM | EC50 |
Mol Endocrinol (2010) 24: 240-9 [PMID:19910453]; Mol Endocrinol (2011) 25: 1040-54 [PMID:21493671] |
| SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745] | ||||||||
| GtoPdb | - | - | 8.8 | pIC50 | - | - | - | Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717] |
| SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346] | ||||||||
| GtoPdb | - | - | 9.8 | pIC50 | - | - | - | Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
