ChEMBL ligand: CHEMBL196478
OT receptor/Oxytocin receptor in Human [ChEMBL: CHEMBL2049] [GtoPdb: 369] [UniProtKB: P30559] There should be some charts here, you may need to enable JavaScript!
V1A receptor/Vasopressin V1a receptor in Human [ChEMBL: CHEMBL1889] [GtoPdb: 366] [UniProtKB: P37288] There should be some charts here, you may need to enable JavaScript!
V1B receptor/Vasopressin V1b receptor in Human [ChEMBL: CHEMBL1921] [GtoPdb: 367] [UniProtKB: P47901] There should be some charts here, you may need to enable JavaScript!
V2 receptor/Vasopressin V2 receptor in Human [ChEMBL: CHEMBL1790] [GtoPdb: 368] [UniProtKB: P30518] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
OT receptor/Oxytocin receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2049] [GtoPdb: 369] [UniProtKB: P30559]
ChEMBL	Displacement of [3H]oxytocin from human OTR	B	8.9	pKi	1.26	nM	Ki	J Med Chem (2006) 49: 4159-4170 [PMID:16821776]
ChEMBL	Binding affinity to human oxytocin receptor	B	8.9	pKi	1.26	nM	Ki	Bioorg Med Chem Lett (2008) 18: 90-94 [PMID:18032036]
ChEMBL	Displacement of [3H]-oxytocin from human oxytocin receptor	B	8.9	pKi	1.26	nM	Ki	J Med Chem (2010) 53: 6525-6538 [PMID:20550119]
GtoPdb	-	-	8.9	pKi	-	-	-	J Med Chem (2005) 48: 6956-69 [PMID:16250654]
V1A receptor/Vasopressin V1a receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1889] [GtoPdb: 366] [UniProtKB: P37288]
ChEMBL	Displacement of [3H]oxytocin from human V1a vasopressin receptor	B	5.2	pKi	<6309.57	nM	Ki	J Med Chem (2005) 48: 6956-6969 [PMID:16250654]
ChEMBL	Displacement of [3H]vasopressin from human vasopressin V1a receptor	B	5.2	pKi	6309.57	nM	Ki	J Med Chem (2010) 53: 6525-6538 [PMID:20550119]
V1B receptor/Vasopressin V1b receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1921] [GtoPdb: 367] [UniProtKB: P47901]
ChEMBL	Displacement of [3H]oxytocin from human V1b vasopressin receptor	B	5.2	pKi	<6309.57	nM	Ki	J Med Chem (2005) 48: 6956-6969 [PMID:16250654]
ChEMBL	Displacement of [3H]vasopressin from human vasopressin V1b receptor	B	5.2	pKi	>6309.57	nM	Ki	J Med Chem (2010) 53: 6525-6538 [PMID:20550119]
V2 receptor/Vasopressin V2 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1790] [GtoPdb: 368] [UniProtKB: P30518]
ChEMBL	Displacement of [3H]oxytocin from human V2 vasopressin receptor	B	6.2	pKi	630.96	nM	Ki	J Med Chem (2005) 48: 6956-6969 [PMID:16250654]
ChEMBL	Displacement of [3H]vasopressin from human vasopressin V2 receptor	B	6.2	pKi	630.96	nM	Ki	J Med Chem (2010) 53: 6525-6538 [PMID:20550119]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]