DY131 [Ligand Id: 2834] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL192509 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Estrogen-related receptor-γ/Estrogen-related receptor gamma in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4245] [GtoPdb: 624] [UniProtKB: P62508] | ||||||||
| ChEMBL | Inhibition of [3H]4-OHT binding to Estrogen-Related Receptor gamma | B | 6.18 | pIC50 | 660 | nM | IC50 | J Med Chem (2005) 48: 3107-3109 [PMID:15857113] |
| GtoPdb | - | - | 6.2 | pIC50 | - | - | - |
Bioorg Med Chem Lett (2005) 15: 1311-3 [PMID:15713377]; J Med Chem (2005) 48: 3107-9 [PMID:15857113] |
| ChEMBL | Estrogen-Related Receptor gamma activity in FRET assay | F | 6.89 | pEC50 | 130 | nM | EC50 | J Med Chem (2005) 48: 3107-3109 [PMID:15857113] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
