ChEMBL ligand: CHEMBL360055 (Gallamine)
Acetylcholinesterase in Torpedo californica [ChEMBL: CHEMBL4780] [UniProtKB: P04058] acetylcholinesterase (Yt blood group)/Acetylcholinesterase in Human [ChEMBL: CHEMBL220] [GtoPdb: 2465] [UniProtKB: P22303] There should be some charts here, you may need to enable JavaScript!
M1 receptor/Muscarinic acetylcholine receptor M1 in Human [ChEMBL: CHEMBL216] [GtoPdb: 13] [UniProtKB: P11229] There should be some charts here, you may need to enable JavaScript!
Muscarinic acetylcholine receptor M2 in Pig [ChEMBL: CHEMBL4781] [UniProtKB: P06199] There should be some charts here, you may need to enable JavaScript!
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172] M2 receptor in Rat [GtoPdb: 14] [UniProtKB: P10980] There should be some charts here, you may need to enable JavaScript!
nicotinic acetylcholine receptor α1 subunit in Human [GtoPdb: 462] [UniProtKB: P02708] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Acetylcholinesterase in Torpedo californica (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4780] [UniProtKB: P04058]
ChEMBL	Inhibition of Torpedo californica AChE	B	4.82	pKi	15000	nM	Ki	J Med Chem (2008) 51: 3154-3170 [PMID:18479118]
acetylcholinesterase (Yt blood group)/Acetylcholinesterase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL220] [GtoPdb: 2465] [UniProtKB: P22303]
ChEMBL	Inhibition of human AChE	B	4.43	pKi	37000	nM	Ki	J Med Chem (2008) 51: 3154-3170 [PMID:18479118]
M1 receptor/Muscarinic acetylcholine receptor M1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL216] [GtoPdb: 13] [UniProtKB: P11229]
ChEMBL	Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in presence of para-LRB-AC42	B	5.07	pKi	8511.38	nM	Ki	J Med Chem (2012) 55: 2125-2143 [PMID:22329602]
Muscarinic acetylcholine receptor M2 in Pig (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4781] [UniProtKB: P06199]
ChEMBL	Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptor	B	6.88	pEC50	131.83	nM	EC50	J Med Chem (2007) 50: 5685-5695 [PMID:17944454]
ChEMBL	Inhibition of [3H]NMS dissociation from porcine muscarinic M2 receptor	B	6.89	pEC50	130	nM	EC50	J Med Chem (2007) 50: 5685-5695 [PMID:17944454]
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172]
GtoPdb	-	-	6.3	pKd	-	-	-	Mol Pharmacol (1995) 48: 362-78 [PMID:7651370]; Br J Pharmacol (1976) 58: 323-31 [PMID:990587]
GtoPdb	-	-	7.6	pKi	-	-	-	J Pharmacol Exp Ther (1998) 284: 500-7 [PMID:9454790]; Mol Pharmacol (2003) 64: 180-90 [PMID:12815174]; Mol Pharmacol (2018) 94: 1298-1309 [PMID:30213802]
M2 receptor in Rat [GtoPdb: 14] [UniProtKB: P10980]
GtoPdb	-	-	5.6	pKi	-	-	-	J Pharmacol Exp Ther (1998) 284: 500-7 [PMID:9454790]
nicotinic acetylcholine receptor α1 subunit in Human [GtoPdb: 462] [UniProtKB: P02708]
GtoPdb	-	-	6	pIC50	~1000	nM	IC50

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]