bantag-1 [Ligand Id: 6176] activity data from GtoPdb

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  • BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336]
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  • BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550]
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  • BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
  • BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
  • BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336]
GtoPdb - - 5.48 pIC50 3300 nM IC50 Cell Metab (2010) 11: 101-12 [PMID:20096642];
Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571]
BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550]
GtoPdb - - 5.36 pIC50 4400 nM IC50 Cell Metab (2010) 11: 101-12 [PMID:20096642];
Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571]
BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
GtoPdb - - 8.7 pIC50 2 nM IC50 Cell Metab (2010) 11: 101-12 [PMID:20096642];
Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571];
J Pharmacol Exp Ther (2019) 369: 454-465 [PMID:30971479]
BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
GtoPdb - - 8.09 pIC50 8.1 nM IC50 Cell Metab (2010) 11: 101-12 [PMID:20096642]
BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
GtoPdb - - 8.77 pIC50 1.7 nM IC50 Cell Metab (2010) 11: 101-12 [PMID:20096642]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.