ChEMBL ligand: CHEMBL597557
coagulation factor IX/Coagulation factor IX in Human [ChEMBL: CHEMBL2016] [GtoPdb: 2364] [UniProtKB: P00740] There should be some charts here, you may need to enable JavaScript!
coagulation factor X/Coagulation factor X in Human [ChEMBL: CHEMBL244] [GtoPdb: 2359] [UniProtKB: P00742] There should be some charts here, you may need to enable JavaScript!
plasminogen activator, urokinase/Urokinase-type plasminogen activator in Human [ChEMBL: CHEMBL3286] [GtoPdb: 2393] [UniProtKB: P00749] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
coagulation factor IX/Coagulation factor IX in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2016] [GtoPdb: 2364] [UniProtKB: P00740]
ChEMBL	Inhibition of human recombinant factor 9a by amidolytic assay	B	8.7	pKi	2	nM	Ki	J Med Chem (2010) 53: 1473-1482 [PMID:20121197]
GtoPdb	-	-	8.7	pIC50	2	nM	IC50	J Med Chem (2010) 53: 1473-82 [PMID:20121197]
coagulation factor X/Coagulation factor X in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL244] [GtoPdb: 2359] [UniProtKB: P00742]
ChEMBL	Inhibition of factor 10a by amidolytic assay	B	6.23	pKi	583	nM	Ki	J Med Chem (2010) 53: 1473-1482 [PMID:20121197]
plasminogen activator, urokinase/Urokinase-type plasminogen activator in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3286] [GtoPdb: 2393] [UniProtKB: P00749]
ChEMBL	Inhibition of uPA	B	6.13	pKi	733	nM	Ki	J Med Chem (2010) 53: 1473-1482 [PMID:20121197]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]