testolactone [Ligand Id: 7303] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1571 (Fludestrin, NSC-23759, SQ 9538, SQ-9538, Teolit, Teslac, Testolactone, Testolactone ciii) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| CYP19A1/Cytochrome P450 19A1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1978] [GtoPdb: 1362] [UniProtKB: P11511] | ||||||||
| ChEMBL | In vitro inhibition of Cytochrome P450 19A1 | B | 4.46 | pKi | 35000 | nM | Ki | J Med Chem (1989) 32: 2231-2239 [PMID:2677377] |
| GtoPdb | - | - | 4.46 | pKi | 35000 | nM | Ki | Cancer Res (1982) 42: 3327s-3333s [PMID:7083195] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
