lixisenatide [Ligand Id: 7387] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL2108336 (Adlyxin, AVE-0010, AVE0010, AVE 010, AVE-010, Lixisenatide, Lyxumia, ZP 10, ZP-10) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220] | ||||||||
| GtoPdb | CHO-K1 cells overexpressing the human GLP-1 receptor. | - | 8.88 | pKi | 1.33 | nM | Ki | Regul Pept (2010) 164: 58-64 [PMID:20570597] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
