compound 34 [PMID: 25974391] [Ligand Id: 8396] activity data from GtoPdb

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  • tripartite motif containing 24 in Human [GtoPdb: 2252] [UniProtKB: O15164]
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  • bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
tripartite motif containing 24 in Human [GtoPdb: 2252] [UniProtKB: O15164]
GtoPdb - - 6.65 pKd 222 nM Kd J Med Chem (2016) 59: 1642-7 [PMID:25974391]
bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
GtoPdb - - 6.86 pKd 137 nM Kd J Med Chem (2016) 59: 1642-7 [PMID:25974391]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.