compound 33 [Toda et al., 2013] [Ligand Id: 8791] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL2409007 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GPR142/Probable G-protein coupled receptor 142 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2069161] [GtoPdb: 132] [UniProtKB: Q7Z601] | ||||||||
| ChEMBL | Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assay | F | 7.66 | pEC50 | 22 | nM | EC50 | ACS Med Chem Lett (2013) 4: 790-794 [PMID:24900747] |
| GtoPdb | - | - | 7.66 | pEC50 | 22 | nM | EC50 | ACS Med Chem Lett (2013) 4: 790-4 [PMID:24900747] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
