4-acryloylphenol [Ligand Id: 8841] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL378577 (4-Acryloylphenol) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 4-aminobutyrate aminotransferase/Gamma-amino-N-butyrate transaminase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2044] [GtoPdb: 2464] [UniProtKB: P80404] | ||||||||
| GtoPdb | - | - | 5.26 | pIC50 | 5480 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-5 [PMID:16290145] |
| ChEMBL | Inhibitory activity against GABAT | B | 5.26 | pIC50 | 5480 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-595 [PMID:16290145] |
| aldehyde dehydrogenase 5 family member A1/Succinate semialdehyde dehydrogenase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1911] [GtoPdb: 2466] [UniProtKB: P51649] | ||||||||
| ChEMBL | Inhibitory activity against SSADH | B | 6.46 | pIC50 | 350 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-595 [PMID:16290145] |
| GtoPdb | - | - | 6.46 | pIC50 | 350 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-5 [PMID:16290145] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
