[111In]DOTA-NOC-ATE

Ligand id: 2064

Name: [111In]DOTA-NOC-ATE    

Classification
Compound class Peptide or derivative
Synonyms
Names References
[111In-DOTA]-NOC-ATE 1
[InIII-DOTA]-NOC-ATE
[InIII-DOTA]-NOC-ATE
Comments
Synthetic radiolabelled peptide. The amino acid sequence of octreotide (SMS 201,995) is modified by replacing the phenylalanine residue at position 3 and C-terminal threoninol with benzoyl-3-thienylalanine and threonine respectively. The peptide is conjugated with DOTA (1,4,7,10-tetraazacyclododecane- 1,4,7,10-tetraacetic acid) and radiolabelled with indium (111I). The structure of the non-radiolabelled version of this ligand is shown in the reference.