triptorelin

Ligand id: 1177

Name: triptorelin

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from ChEMBL and GtoPdb across species (New!)

Selectivity at human GPCRs
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Target Type Action Affinity Units Concentration range (M) Reference
GnRH1 receptor Agonist Full agonist 9.3 – 9.5 pKi - 1
pKi 9.3 – 9.5 (Ki 5.1x10-10 – 3.2x10-10 M) [1]
Selectivity at rat GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
GnRH1 receptor Agonist Full agonist 8.5 – 8.8 pKi - 1
pKi 8.5 – 8.8 [1]