[Phe13,Tyr19]MCH   Click here for help

GtoPdb Ligand ID: 1297

Synonyms: [Phe13,Tyr19]-melanin-concentrating hormone
Comment: Synthetic analogue of MCH
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
MCH1 receptor Rn Agonist Full agonist 9.2 – 9.5 pKi - 4
pKi 9.2 – 9.5 [4]
MCH1 receptor Hs Agonist Full agonist 8.2 – 10.0 pIC50 - 1-3
pIC50 8.2 – 10.0 [1-3]
MCH2 receptor Hs Agonist Full agonist 8.4 – 9.2 pIC50 - 3,5
pIC50 8.4 – 9.2 [3,5]