HS024   Click here for help

GtoPdb Ligand ID: 1328

Synonyms: cyclic[AcCys3,Nle4,Arg5,D-Nal7,Cys-NH2(11)]alpha-MSH-(3-11) | HS 024
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
MC4 receptor Hs Antagonist Antagonist 9.5 pKd - 1
pKd 9.5 [1]
MC5 receptor Hs Antagonist Antagonist 8.5 pKd - 1
pKd 8.5 [1]
MC3 receptor Hs Antagonist Antagonist 8.3 pKd - 1
pKd 8.3 [1]
MC1 receptor Hs Antagonist Antagonist 7.7 pKd - 1
pKd 7.7 [1]