L-362,855   Click here for help

GtoPdb Ligand ID: 2014

Synonyms: L 362855 | L-362855
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 8.4 – 8.8 pKi - 3-5
pKi 8.4 – 8.8 [3-5]
SST5 receptor Hs Agonist Full agonist 7.2 – 9.2 pKi - 2-5
pKi 7.2 – 9.2 [2-5]
SST5 receptor Mm Agonist Full agonist 7.7 – 8.7 pKi - 1
pKi 7.7 – 8.7 [1]
SST3 receptor Hs Agonist Full agonist 7.6 – 8.3 pKi - 3,5
pKi 7.6 – 8.3 [3,5]
SST2 receptor Rn Agonist Full agonist 7.9 pKi - 2
pKi 7.9 [2]
SST2 receptor Mm Agonist Full agonist 7.0 – 8.5 pKi - 2
pKi 7.0 – 8.5 [2]
SST5 receptor Rn Agonist Full agonist 7.3 pKi - 2
pKi 7.3 [2]
SST4 receptor Hs Agonist Full agonist 6.8 – 7.3 pKi - 3,5
pKi 6.8 – 7.3 [3,5]
SST1 receptor Hs Agonist Full agonist 6.1 – 6.2 pKi - 3,5
pKi 6.1 – 6.2 [3,5]