[L-Tyr8]CYN 154806   Click here for help

GtoPdb Ligand ID: 2029

Synonyms: cyanamid 154806
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Antagonist Antagonist 8.1 – 8.4 pKi - 2
pKi 8.1 – 8.4 [2]
SST5 receptor Hs Antagonist Antagonist 7.3 – 9.1 pKi - 2
pKi 7.3 – 9.1 [2]
SST5 receptor Mm Antagonist Antagonist 6.2 – 7.2 pKi - 1
pKi 6.2 – 7.2 [1]
SST3 receptor Hs Antagonist Antagonist 6.2 – 6.8 pKi - 1
pKi 6.2 – 6.8 [1]
SST4 receptor Hs Antagonist Antagonist 6.2 – 6.5 pKi - 2
pKi 6.2 – 6.5 [2]
SST1 receptor Hs Antagonist Antagonist 5.7 – 5.9 pKi - 2
pKi 5.7 – 5.9 [2]