octreotide

Ligand id: 2055

Name: octreotide

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from ChEMBL and GtoPdb across species (New!)

Selectivity at human GPCRs
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Target Type Action Affinity Units Concentration range (M) Reference
SST2 receptor Agonist Full agonist 8.7 – 9.9 pKi - 1,5,7-10
pKi 8.7 – 9.9 [1,5,7-10]
SST5 receptor Agonist Full agonist 7.2 – 9.5 pKi - 1,4-5,7-10
pKi 7.2 – 9.5 [1,4-5,7-10]
SST3 receptor Agonist Full agonist 7.4 – 8.6 pKi - 1-2,5,7,9-10
pKi 7.4 – 8.6 [1-2,5,7,9-10]
Selectivity at mouse GPCRs
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Target Type Action Affinity Units Concentration range (M) Reference
SST5 receptor Agonist Full agonist 7.7 – 9.9 pKi - 3
pKi 7.7 – 9.9 [3]
SST2 receptor Agonist Full agonist 7.5 – 9.2 pKi - 4
pKi 7.5 – 9.2 [4]
SST3 receptor Agonist Full agonist 8.5 pIC50 - 6
pIC50 8.5 [6]
Selectivity at rat GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
SST2 receptor Agonist Full agonist 8.7 pKi - 4
pKi 8.7 [4]
SST3 receptor Agonist Full agonist 7.8 pKi - 4
pKi 7.8 [4]
SST5 receptor Agonist Full agonist 7.8 pKi - 4
pKi 7.8 [4]