• Home
• About »
  • About The Guide to Pharmacology
  • Sponsors
  • Citing
  • Disclaimer
  • Privacy and Cookie Policy
• GRAC database »
  • GPCRs
  • Ion channels »
    • LGICs
    • VGICs
    • Other channels
  • Nuclear receptors
  • Catalytic receptors
  • Transporters
  • Enzymes
  • GRAC editors
  • GRAC consultants
• IUPHAR database
• Ligands »
  • Ligand list
  • Ligand search
• Resources »
  • Help
  • GRAC tutorial
  • GRAC 5th edition HTML
  • GRAC 5th edition PDF
  • Publications
• Advanced search »
  • Target search
  • Ligand search

Selectivity data from the Guide to Receptors and Channels (GRAC), 5th Edition. Selectivity at human targets (unless otherwise stated) Key to terms and symbols Click column headers to sort Receptor Type Action Affinity Units Concentration range (M) Reference V1B receptor Agonist Full agonist 9.0 – 9.7 pKi - 1-2 Selectivity data from IUPHAR-DB Selectivity at human GPCRs Key to terms and symbols Click column headers to sort Receptor Type Action Affinity Units Concentration range (M) Reference V1B receptor Agonist Full agonist 9.0 – 9.7 pKi - 1-2 OT receptor Agonist Full agonist 7.1 – 7.7 pKi - 1-2 V1A receptor Agonist Full agonist 7.1 pKi - 1 V2 receptor Agonist Full agonist 6.5 pKi - 1 Please note: The activity data given on this ligand page represents selected literature values and may not include all reported data. For more details please contact: curators@iuphar-db.org

Disclaimer: Peptide pages are currently under development, please exercise caution over the use of sequence and structural information provided here. Please send notification of errors to curators@iuphar-db.org.