atosiban

Ligand id: 2213

Name: atosiban

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Affinity Units Concentration range (M) Reference
V1A receptor Hs Antagonist Antagonist 8.3 – 8.5 pKi - 1-2,5-6
pKi 8.3 – 8.5 [1-2,5-6]
OT receptor Rn Antagonist Antagonist 7.1 pKi - 2
pKi 7.1 [2]
OT receptor Hs Antagonist Antagonist 6.0 – 7.6 pKi - 1-2,4-6
pKi 6.0 – 7.6 [1-2,4-6]
V1B receptor Hs Antagonist Antagonist 6.2 – 6.6 pKi - 2,6
pKi 6.2 – 6.6 [2,6]
V2 receptor Hs Antagonist Antagonist 5.5 – 6.0 pKi - 2,6
pKi 5.5 – 6.0 [2,6]