atosiban

Ligand id: 2213

Name: atosiban

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from ChEMBL and GtoPdb across species (New!)

Selectivity at human GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
V1A receptor Antagonist Antagonist 8.3 – 8.5 pKi - 1-2,5-6
pKi 8.3 – 8.5 [1-2,5-6]
OT receptor Antagonist Antagonist 6.0 – 7.6 pKi - 1-2,4-6
pKi 6.0 – 7.6 [1-2,4-6]
V1B receptor Antagonist Antagonist 6.2 – 6.6 pKi - 2,6
pKi 6.2 – 6.6 [2,6]
V2 receptor Antagonist Antagonist 5.5 – 6.0 pKi - 2,6
pKi 5.5 – 6.0 [2,6]
Selectivity at rat GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
OT receptor Antagonist Antagonist 7.1 pKi - 2
pKi 7.1 [2]