buserelin

Ligand id: 3860

Name: buserelin

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from ChEMBL and GtoPdb across species (New!)

Selectivity at human GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
GnRH1 receptor Agonist Full agonist 9.5 – 10.4 pKd - 1
pKd 9.5 – 10.4 (Kd 3x10-10 – 4x10-11 M) [1]
GnRH1 receptor Agonist Full agonist 9.4 – 10.0 pKi - 1
pKi 9.4 – 10.0 (Ki 4x10-10 – 1x10-10 M) [1]
GnRH1 receptor Agonist Full agonist 10.5 pEC50 - 2
pEC50 10.5 (EC50 3x10-11 M) [2]
Selectivity at mouse GPCRs
Key to terms and symbols Click column headers to sort
Target Type Action Affinity Units Concentration range (M) Reference
GnRH1 receptor Agonist Full agonist 9.3 – 10.1 pEC50 - 2
pEC50 9.3 – 10.1 (EC50 4.6x10-10 – 9x10-11 M) [2]