buserelin

Ligand id: 3860

Name: buserelin

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Affinity Units Concentration range (M) Reference
GnRH1 receptor Hs Agonist Full agonist 9.5 – 10.4 pKd - 1
pKd 9.5 – 10.4 (Kd 3x10-10 – 4x10-11 M) [1]
GnRH1 receptor Hs Agonist Full agonist 9.4 – 10.0 pKi - 1
pKi 9.4 – 10.0 (Ki 4x10-10 – 1x10-10 M) [1]
GnRH1 receptor Hs Agonist Full agonist 10.5 pEC50 - 2
pEC50 10.5 (EC50 3x10-11 M) [2]
GnRH1 receptor Mm Agonist Full agonist 9.3 – 10.1 pEC50 - 2
pEC50 9.3 – 10.1 (EC50 4.6x10-10 – 9x10-11 M) [2]