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2D Structure

Selectivity data from the Guide to Receptors and Channels (GRAC), 5th Edition. Selectivity at human targets (unless otherwise stated) Key to terms and symbols Click column headers to sort Receptor Type Action Affinity Units Concentration range (M) Reference α3 (α3β2) Antagonist Antagonist - - - α5 Antagonist Antagonist - - - α6 (α6β2*) Antagonist Antagonist - - - Please note: The activity data given on this ligand page represents selected literature values and may not include all reported data. For more details please contact: curators@iuphar-db.org

Disclaimer: Peptide pages are currently under development, please exercise caution over the use of sequence and structural information provided here. Please send notification of errors to curators@iuphar-db.org.