|
|
|
A1 receptor
|
|
|
Rn |
Agonist |
Agonist |
8.9 |
pKi |
- |
4 |
|
⤷ |
pKi
8.9
(Ki 1.2x10-9 M)
[4]
|
A3 receptor
|
|
|
Hs |
Agonist |
Full agonist |
7.1 – 8.1 |
pKi |
- |
6-7,11,16,19 |
|
⤷ |
pKi
7.1 – 8.1
[6-7,11,16,19]
|
A1 receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.4 – 8.7 |
pKi |
- |
6,9,11,15,17 |
|
⤷ |
pKi
6.4 – 8.7
[6,9,11,15,17]
|
A3 receptor
|
|
|
Rn |
Agonist |
Full agonist |
6.6 – 6.8 |
pKi |
- |
4,14 |
|
⤷ |
pKi
6.6 – 6.8
[4,14]
|
A2A receptor
|
|
|
Rn |
Agonist |
Agonist |
6.7 |
pKi |
- |
4 |
|
⤷ |
pKi
6.7
(Ki 2.2x10-7 M)
[4]
|
A2A receptor
|
|
|
Hs |
Agonist |
Full agonist |
6.0 – 6.2 |
pKi |
- |
5-6,10-12 |
|
⤷ |
pKi
6.0 – 6.2
[5-6,10-12]
|
A2B receptor
|
|
|
Mm |
Agonist |
Agonist |
4.7 |
pKi |
- |
2 |
|
⤷ |
pKi
4.7
(Ki 1.9x10-5 M)
[2]
|
A2B receptor
|
|
|
Hs |
Agonist |
Full agonist |
3.8 – 5.5 |
pKi |
- |
1,3,8,13,18 |
|
⤷ |
pKi
3.8 – 5.5
[1,3,8,13,18]
|
|