demotate 2   Click here for help

GtoPdb Ligand ID: 5636

Synonyms: N(4) (0-1),Asp0,Tyr3-octreotate
Comment: Demotate 2 can be radiolabelled with 99mTechnetium, a metastable nuclear isomer of Technetium-99 and is widely used in diagnostic nuclear medicine.
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Hs Agonist Full agonist 8.5 pIC50 - 1
pIC50 8.5 (IC50 3.2x10-9 M) [1]