icatibant

Ligand id: 667

Name: icatibant

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Affinity Units Concentration range (M) Reference
B2 receptor Hs Antagonist Antagonist 8.4 pA2 - 6
pA2 8.4 [6]
B2 receptor Hs Antagonist Antagonist 10.2 pKi - 1
pKi 10.2 (Ki 6.4x10-11 M) [1]
B2 receptor Rn Antagonist Antagonist 10.0 – 10.3 pKi - 4
pKi 10.0 – 10.3 [4]
B2 receptor Mm Antagonist Antagonist 9.6 pKi - 7
pKi 9.6 [7]
B1 receptor Hs Antagonist Antagonist 6.4 – 7.0 pKi - 3,8
pKi 6.4 – 7.0 [3,8]
B1 receptor Rn Antagonist Antagonist 6.1 – 6.4 pKi - 8
pKi 6.1 – 6.4 [8]
B2 receptor Hs Antagonist Antagonist 8.0 – 9.4 pIC50 - 2,7
pIC50 8.0 – 9.4 [2,7]