histerelin   Click here for help

GtoPdb Ligand ID: 9344

Comment: GnRH agonist peptide
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
GnRH1 receptor Hs Agonist Full agonist 9.0 – 10.4 pKd - 1
pKd 9.0 – 10.4 (Kd 1x10-9 – 4x10-11 M) [1]
GnRH1 receptor Hs Agonist Full agonist 8.7 – 9.7 pKi - 1
pKi 8.7 – 9.7 (Ki 1.9x10-9 – 2x10-10 M) [1]