AY77   Click here for help

GtoPdb Ligand ID: 9455

Synonyms: compound 14 [PMID: 26819675]
Comment: AY77 is a potent small molecule, peptidic PAR2 agonist [1]. The compound is stable in rat plasma making it suitable for physiological studies.
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
PAR2 Hs Agonist Agonist 7.5 pEC50 - 1
pEC50 7.5 (EC50 3.3x10-8 M) [1]