resiniferatoxin

Ligand id: 2491

Name: resiniferatoxin

Abbreviated name: RTX

Structure and Physico-chemical Properties

2D Structure
Calculated Physico-chemical Properties
Hydrogen bond acceptors 7
Hydrogen bond donors 2
Rotatable bonds 9
Topological polar surface area 120.75
Molecular weight 628.27
XLogP 2.85
No. Lipinski's rules broken 0

Molecular properties generated using the CDK

References
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Cloning and pharmacological characterization of mouse TRPV1.
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Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
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The vanilloid agonist resiniferatoxin for interventional-based pain control.
Curr Top Med Chem, 11 (17): 2171-9. [PMID:21671877]
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