buserelin

Ligand id: 3860

Name: buserelin

Structure and Physico-chemical Properties

2D Structure
Classification
Compound class Peptide or derivative
Approved drug? Yes
IUPAC Name
(2S)-N-[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S)-1-[[(2S)-5-(diaminomethylideneamino)-1-[(2S)-2-(ethylcarbamoyl)pyrrolidin-1-yl]-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-[(2-methylpropan-2-yl)oxy]-1-oxopropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-(3H-imidazol-4-yl)-1-oxopropan-2-yl]-5-oxopyrrolidine-2-carboxamide
International Nonproprietary Names
INN number INN
4045 buserelin
Synonyms
buserelin acetate | HOE 766 | HOE 766A | ICI 123215 | Metrelef® | Suprefact®
Database Links
CAS Registry No. 57982-77-1 (source: Scifinder)
ChEMBL Ligand CHEMBL2110824
DrugBank Ligand DB06719
GtoPdb PubChem SID 178100699
PubChem CID 50225
Search Google for chemical match using the InChIKey CUWODFFVMXJOKD-UVLQAERKSA-N
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Search UniChem for chemical match using the InChIKey CUWODFFVMXJOKD-UVLQAERKSA-N
Search UniChem for chemicals with the same backbone CUWODFFVMXJOKD
Wikipedia Buserelin
Comments
Buserelin is a GnRH (luteinizing hormone-releasing hormone, LHRH) agonist. Buserelin does not appear to have marketing approval for human use in the US or EU, although individual countries may have approved use of this drug.