bromodomain and PHD finger containing 3 | Non-enzymatic BRD containing proteins | IUPHAR/BPS Guide to PHARMACOLOGY

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bromodomain and PHD finger containing 3

Target not currently curated in GtoImmuPdb

Target id: 2731

Nomenclature: bromodomain and PHD finger containing 3

Family: Non-enzymatic BRD containing proteins

Annotation status:  image of a grey circle Awaiting annotation/under development. Please contact us if you can help with annotation.  » Email us

Gene and Protein Information
Species TM AA Chromosomal Location Gene Symbol Gene Name Reference
Human - 1205 6p21.31 BRPF3 bromodomain and PHD finger containing 3
Mouse - 1204 17 A3.3 Brpf3 bromodomain and PHD finger containing
Rat - 1199 20p12 Brpf3 bromodomain and PHD finger containing
Previous and Unofficial Names
bromodomain and PHD finger containing, 3 | bromodomain and PHD finger containing
Database Links
CATH/Gene3D
ChEMBL Target
Ensembl Gene
Entrez Gene
Human Protein Atlas
KEGG Gene
RefSeq Nucleotide
RefSeq Protein
UniProtKB
Wikipedia
Other Binding Ligands
Key to terms and symbols Click column headers to sort
Ligand Sp. Action Affinity Parameter Reference
NI-57 Hs Binding 6.4 pKd 2
pKd 6.4 (Kd 4.08x10-7 M) [2]
OF-1 Hs Binding 5.6 pKd 1
pKd 5.6 (Kd 2.4x10-6 M) [1]
Description: By isothermal titration calorimetry.

References

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1. SGC. OF-1 A chemical probe for BRPF bromodomains. Accessed on 05/04/2017. Modified on 05/04/2017. SGC, http://www.thesgc.org/chemical-probes/OF-1

2. Structural Genomics Consortium. NI-57 – a chemical probe for BRPF bromodomains. Accessed on 15/07/2015. Modified on 15/07/2015. http://www.thesgc.org, http://www.thesgc.org/chemical-probes/NI-57

How to cite this page

Non-enzymatic BRD containing proteins: bromodomain and PHD finger containing 3. Last modified on 05/04/2017. Accessed on 23/04/2019. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2731.