target,target_id,target_uniprot,target_species,ligand,ligand_id,ligand_species,ligand_pubchem_cid,smiles,inchi,inchikey,type,action,action_comment,endogenous,primary_target,concentration_range,affinity_parameter,affinity_high,affinity_median,affinity_low,original_affinity_units,original_affinity_low_nm,original_affinity_median_nm,original_affinity_high_nm,original_affinity_relation,assay_description,receptor_site,ligand_context,pubmed_id FZD8,236,Q9H461,Human,carbamazepine,5339,,2554,NC(=O)N1c2ccccc2C=Cc2c1cccc2,"InChI=1S/C15H12N2O/c16-15(18)17-13-7-3-1-5-11(13)9-10-12-6-2-4-8-14(12)17/h1-10H,(H2,16,18)",FFGPTBGBLSHEPO-UHFFFAOYSA-N,Allosteric modulator,Negative,,,,,pKd,,4.77,,Kd,,16800.0,,=,Binding affinity for FZD8 cysteine-rich domain (CRD) by SPR analysis.,,,32049522, FZD8,236,Q9H461,Human,vantictumab,10197,,,,,,Antibody,Antagonist,,,,,pIC50,,8.0,,IC50,,10.0,,~,,,,22753465,