target,target_id,target_uniprot,target_species,ligand,ligand_id,ligand_species,ligand_pubchem_cid,smiles,inchi,inchikey,type,action,action_comment,endogenous,primary_target,concentration_range,affinity_parameter,affinity_high,affinity_median,affinity_low,original_affinity_units,original_affinity_low_nm,original_affinity_median_nm,original_affinity_high_nm,original_affinity_relation,assay_description,receptor_site,ligand_context,pubmed_id CX3CR1,74,P49238,Human,CX3CL1,856,Human,,,,,Agonist,Full agonist,,yes,,,pIC50,,8.9,,,,,,=,,,,14607932, CX3CR1,74,P49238,Human,JMS-17-2,10390,,57382073,Clc1ccc(cc1)C1CCN(CC1)CCCn1c(=O)c2cccn2c2c1cccc2,"InChI=1S/C25H26ClN3O/c26-21-10-8-19(9-11-21)20-12-17-27(18-13-20)14-4-16-29-23-6-2-1-5-22(23)28-15-3-7-24(28)25(29)30/h1-3,5-11,15,20H,4,12-14,16-18H2",WOSMCMULWWHMIV-UHFFFAOYSA-N,Antagonist,Antagonist,,,,,pIC50,,9.49,,IC50,,0.32,,=,Measuring the inhibition of FKN-stimulated ERK1/2 phosphorylation.,,,27001765,