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A list of approved drugs that modulate GABAA channel activity by binding to the allosteric benzodiazepine site. These drugs increase the inhibitory effects of GABA.
alprazolam
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chlordiazepoxide
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clobazam
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clonazepam
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clorazepate
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diazepam
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estazolam
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eszopiclone
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flumazenil
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flunitrazepam
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flurazepam
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halazepam
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lorazepam
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lormetazepam
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midazolam
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oxazepam
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quazepam
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temazepam
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triazolam
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zaleplon
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zolpidem
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Database page citation:
Benzodiazepine class drugs. Accessed on 17/02/2025. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=1072.