CDK12 inhibitor 2 [Ligand Id: 10063] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| cyclin dependent kinase 12 in Human [GtoPdb: 1965] [UniProtKB: Q9NYV4] | ||||||||
| GtoPdb | - | - | 7.28 | pIC50 | 52 | nM | IC50 | J Med Chem (2018) 61: 7710-7728 [PMID:30067358] |
| cyclin dependent kinase 13 in Human [GtoPdb: 1966] [UniProtKB: Q14004] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | 10 | nM | IC50 | J Med Chem (2018) 61: 7710-7728 [PMID:30067358] |
| cyclin dependent kinase 7 in Human [GtoPdb: 1979] [UniProtKB: P50613] | ||||||||
| GtoPdb | - | - | 5 | pIC50 | >10000 | nM | IC50 | J Med Chem (2018) 61: 7710-7728 [PMID:30067358] |
| cyclin dependent kinase 8 in Human [GtoPdb: 1980] [UniProtKB: P49336] | ||||||||
| GtoPdb | - | - | 5 | pIC50 | >10000 | nM | IC50 | J Med Chem (2018) 61: 7710-7728 [PMID:30067358] |
| cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750] | ||||||||
| GtoPdb | - | - | 4.8 | pIC50 | 16000 | nM | IC50 | J Med Chem (2018) 61: 7710-7728 [PMID:30067358] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
