Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
kelch like ECH-associated protein 1 in Human [GtoPdb: 2757] [UniProtKB: Q14145] | ||||||||
GtoPdb | Binding to hKEAP1 by SPR. | - | 6.99 | pKd | 102 | nM | Kd | J Med Chem (2018) 61: 8029-8047 [PMID:30122040] |
GtoPdb | Measured by fluorescence anisotropy. | - | 7.22 | pIC50 | 60 | nM | IC50 | J Med Chem (2018) 61: 8029-8047 [PMID:30122040] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.