acalisib [Ligand Id: 10096] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | In an in vitro biochemical assay using recombinant enzyme. | - | 5.26 | pIC50 | 5441 | nM | IC50 | J Biol Chem (2013) 288: 35346-57 [PMID:24133210] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | In an in vitro biochemical assay using recombinant enzyme. | - | 5.47 | pIC50 | 3377 | nM | IC50 | J Biol Chem (2013) 288: 35346-57 [PMID:24133210] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | In an in vitro biochemical assay using recombinant enzyme. | - | 7.9 | pIC50 | 12.7 | nM | IC50 | J Biol Chem (2013) 288: 35346-57 [PMID:24133210] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | In an in vitro biochemical assay using recombinant enzyme. | - | 5.86 | pIC50 | 1389 | nM | IC50 | J Biol Chem (2013) 288: 35346-57 [PMID:24133210] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
