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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
neurotrophic receptor tyrosine kinase 1 in Human [GtoPdb: 1817] [UniProtKB: P04629] | ||||||||
GtoPdb | - | - | 7 | pKd | 100 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
neurotrophic receptor tyrosine kinase 2 in Human [GtoPdb: 1818] [UniProtKB: Q16620] | ||||||||
GtoPdb | - | - | 7.96 | pKd | 11 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
neurotrophic receptor tyrosine kinase 3 in Human [GtoPdb: 1819] [UniProtKB: Q16288] | ||||||||
GtoPdb | - | - | 8.03 | pKd | 9.3 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
EPH receptor A2 in Human [GtoPdb: 1822] [UniProtKB: P29317] | ||||||||
GtoPdb | - | - | 6.59 | pKd | 260 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
EPH receptor A7 in Human [GtoPdb: 1827] [UniProtKB: Q15375] | ||||||||
GtoPdb | - | - | 6.7 | pKd | 200 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
EPH receptor A8 in Human [GtoPdb: 1828] [UniProtKB: P29322] | ||||||||
GtoPdb | - | - | 7.1 | pKd | 79 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
EPH receptor B2 in Human [GtoPdb: 1831] [UniProtKB: P29323] | ||||||||
GtoPdb | - | - | 6.59 | pKd | 260 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
TEK receptor tyrosine kinase in Human [GtoPdb: 1842] [UniProtKB: Q02763] | ||||||||
GtoPdb | - | - | 6.43 | pKd | 370 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
discoidin domain receptor tyrosine kinase 1 in Human [GtoPdb: 1843] [UniProtKB: Q08345] | ||||||||
GtoPdb | - | - | 8.1 | pKd | 7.9 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
GtoPdb | - | - | 8.03 | pIC50 | 9.4 | nM | IC50 | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
discoidin domain receptor tyrosine kinase 2 in Human [GtoPdb: 1844] [UniProtKB: Q16832] | ||||||||
GtoPdb | - | - | 8.1 | pKd | 8 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
GtoPdb | - | - | 7.69 | pIC50 | 20.4 | nM | IC50 | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
ABL proto-oncogene 1, non-receptor tyrosine kinase in Human [GtoPdb: 1923] [UniProtKB: P00519] | ||||||||
GtoPdb | - | - | 6.31 | pIC50 | 494 | nM | IC50 | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
GtoPdb | - | - | 6.74 | pKd | 180 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
serine/threonine kinase 10 in Human [GtoPdb: 2211] [UniProtKB: O94804] | ||||||||
GtoPdb | - | - | 8 | pKd | 10 | nM | Kd | J Med Chem (2018) 61: 7977-7990 [PMID:30075624] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.