TUG-1375 [Ligand Id: 10107] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| FFA2 receptor in Human [GtoPdb: 226] [UniProtKB: O15552] | ||||||||
| GtoPdb | Binding affinity for hFFA2. | - | 6.69 | pKi | 204 | nM | Ki | J Med Chem (2018) 61: 9534-9550 [PMID:30247908] |
| GtoPdb | Agonist activity in a BRET-based β-arrestin-2 recruitment assay. | - | 6.1 | pEC50 | 794 | nM | EC50 | J Med Chem (2018) 61: 9534-9550 [PMID:30247908] |
| GtoPdb | Agonist activity in a cAMP inhibition assay. | - | 7.11 | pEC50 | 77.6 | nM | EC50 | J Med Chem (2018) 61: 9534-9550 [PMID:30247908] |
| FFA2 receptor in Mouse [GtoPdb: 226] [UniProtKB: Q8VCK6] | ||||||||
| GtoPdb | - | - | 6.44 | pEC50 | 363 | nM | EC50 | J Med Chem (2018) 61: 9534-9550 [PMID:30247908] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
