GSK2646264 [Ligand Id: 10108] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 4.5 | pIC50 | 31622 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| aurora kinase A in Human [GtoPdb: 1936] [UniProtKB: O14965] | ||||||||
| GtoPdb | - | - | 4.3 | pIC50 | >50119 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| aurora kinase B in Human [GtoPdb: 1937] [UniProtKB: Q96GD4] | ||||||||
| GtoPdb | - | - | 4.6 | pIC50 | >25119 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| glycogen synthase kinase 3 beta in Human [GtoPdb: 2030] [UniProtKB: P49841] | ||||||||
| GtoPdb | - | - | 5.3 | pIC50 | 5012 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 5 | pIC50 | 10000 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
| GtoPdb | - | - | 5.4 | pIC50 | 3981 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| leucine rich repeat kinase 2 in Human [GtoPdb: 2059] [UniProtKB: Q5S007] | ||||||||
| GtoPdb | - | - | 5.4 | pIC50 | 3981 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
| spleen associated tyrosine kinase in Human [GtoPdb: 2230] [UniProtKB: P43405] | ||||||||
| GtoPdb | - | - | 7.1 | pIC50 | 79.4 | nM | IC50 | Bioorg Med Chem Lett (2018) 28: 3458-3462 [PMID:30249354] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
