compound 27d [PMID: 28231433] [Ligand Id: 10218] activity data from GtoPdb

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  • sphingosine kinase 1 in Human [GtoPdb: 2204] [UniProtKB: Q9NYA1]
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  • sphingosine kinase 2 in Human [GtoPdb: 2205] [UniProtKB: Q9NRA0]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
sphingosine kinase 1 in Human [GtoPdb: 2204] [UniProtKB: Q9NYA1]
GtoPdb - - 5.01 pIC50 9820 nM IC50 J Med Chem (2017) 60: 2562-2572 [PMID:28231433]
sphingosine kinase 2 in Human [GtoPdb: 2205] [UniProtKB: Q9NRA0]
GtoPdb - - 6.84 pIC50 145 nM IC50 J Med Chem (2017) 60: 2562-2572 [PMID:28231433]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.