LEI105 [Ligand Id: 10246] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| diacylglycerol lipase α in Human [GtoPdb: 1396] [UniProtKB: Q9Y4D2] | ||||||||
| GtoPdb | - | - | 7.89 | pIC50 | 13 | nM | IC50 | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
| GtoPdb | Inhibition of recombinant human DAGα in a biochemical assay with para-nitrophenylbutyrate as a surrogate substrate. | - | 8.5 | pIC50 | - | - | - | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
| diacylglycerol lipase β in Human [GtoPdb: 1397] [UniProtKB: Q8NCG7] | ||||||||
| GtoPdb | Inhibition of recombinant human DAGβ in a biochemical assay with para-nitrophenylbutyrate as a surrogate substrate. | - | 8.1 | pIC50 | - | - | - | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
