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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| B-Raf proto-oncogene, serine/threonine kinase in Human [GtoPdb: 1943] [UniProtKB: P15056] | ||||||||
| GtoPdb | Determined in a Latha screen assay. | - | 6.49 | pIC50 | 322 | nM | IC50 | Br J Pharmacol (2019) 176: 2095-2108 [PMID:30825190] |
| receptor interacting serine/threonine kinase 1 in Human [GtoPdb: 2189] [UniProtKB: Q13546] | ||||||||
| GtoPdb | Determined in a KINOMEscan assay. | - | 7.01 | pKd | 97 | nM | Kd | Br J Pharmacol (2019) 176: 2095-2108 [PMID:30825190] |
| receptor interacting serine/threonine kinase 3 in Human [GtoPdb: 2191] [UniProtKB: Q9Y572] | ||||||||
| GtoPdb | Determined in a KINOMEscan assay. | - | 7.11 | pKd | 77 | nM | Kd | Br J Pharmacol (2019) 176: 2095-2108 [PMID:30825190] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.