compound 23 [PMID: 31398032] [Ligand Id: 10445] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ATPase family AAA domain containing 2 in Human [GtoPdb: 2719] [UniProtKB: Q6PL18] | ||||||||
| GtoPdb | Measuring small-molecule competition using TR-FRET assay with ATAD2 construct 6 (Flag-6H-tev-ATAd2(981-1121) and the biotinylated triacetylated histone H4 peptide (SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGAKRHRKV-biotin). | - | 6.5 | pIC50 | 316 | nM | IC50 | J Med Chem (2019) 62: 7506-7525 [PMID:31398032] |
| ATPase family AAA domain containing 2B in Human [GtoPdb: 2720] [UniProtKB: Q9ULI0] | ||||||||
| GtoPdb | Measuring small-molecule competition using TR-FRET assay with ATAD2 construct 6 (Flag-6H-tev-ATAd2(981-1121) and the biotinylated triacetylated histone H4 peptide (SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGAKRHRKV-biotin). | - | 6.3 | pIC50 | 501 | nM | IC50 | J Med Chem (2019) 62: 7506-7525 [PMID:31398032] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
