dBET6 [Ligand Id: 10534] activity data from GtoPdb

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  • bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 4 in Human [GtoPdb: 1945] [UniProtKB: O60885]
GtoPdb Inhibition of BRD4 (BD1) kinase activity. - 7.85 pIC50 14 nM IC50 Mol Cell (2017) 67: 5-18.e19 [PMID:28673542]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.