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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
ribosomal protein S6 kinase A6 in Human [GtoPdb: 1530] [UniProtKB: Q9UK32] | ||||||||
GtoPdb | - | - | 6.56 | pIC50 | 276 | nM | IC50 | J Med Chem (2020) 63: 601-612 [PMID:31859507] |
fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888] | ||||||||
GtoPdb | - | - | 6.91 | pIC50 | 123 | nM | IC50 | J Med Chem (2020) 63: 601-612 [PMID:31859507] |
inhibitor of nuclear factor kappa B kinase subunit epsilon in Human [GtoPdb: 2040] [UniProtKB: Q14164] | ||||||||
GtoPdb | - | - | 8.7 | pIC50 | 2 | nM | IC50 | J Med Chem (2020) 63: 601-612 [PMID:31859507] |
serine/threonine kinase 17a in Human [GtoPdb: 2214] [UniProtKB: Q9UEE5] | ||||||||
GtoPdb | - | - | 6.51 | pIC50 | 311 | nM | IC50 | J Med Chem (2020) 63: 601-612 [PMID:31859507] |
TANK binding kinase 1 in Human [GtoPdb: 2237] [UniProtKB: Q9UHD2] | ||||||||
GtoPdb | Inhibition at low ATP concentration. | - | 8.7 | pIC50 | 2 | nM | IC50 | J Med Chem (2020) 63: 601-612 [PMID:31859507] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.