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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143] | ||||||||
| GtoPdb | Competitive membrane binding assay measuring displacement [3H]DPDPE from human δ receptors expressed by CHO cells. | - | 5.38 | pKi | 4150 | nM | Ki | J Pharmacol Exp Ther (2017) 363: 104-113 [PMID:28778859] |
| μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
| GtoPdb | Competitive membrane binding assay measuring displacement [3H]naloxone from human μ receptors expressed by CHO cells. | - | 6.63 | pKi | 237 | nM | Ki | J Pharmacol Exp Ther (2017) 363: 104-113 [PMID:28778859] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.