BMS-986260 [Ligand Id: 10662] activity data from GtoPdb

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  • activin A receptor type 1 in Human [GtoPdb: 1785] [UniProtKB: Q04771]
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  • activin A receptor type 1B in Human [GtoPdb: 1787] [UniProtKB: P36896]
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  • transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
activin A receptor type 1 in Human [GtoPdb: 1785] [UniProtKB: Q04771]
GtoPdb - - 7.15 pIC50 70.4 nM IC50 ACS Med Chem Lett (2020) 11: 172-178 [PMID:32071685]
activin A receptor type 1B in Human [GtoPdb: 1787] [UniProtKB: P36896]
GtoPdb - - 7.48 pIC50 33.3 nM IC50 ACS Med Chem Lett (2020) 11: 172-178 [PMID:32071685]
transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897]
GtoPdb - - 8.8 pIC50 1.6 nM IC50 ACS Med Chem Lett (2020) 11: 172-178 [PMID:32071685]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.