UCSF3384 [Ligand Id: 10665] activity data from GtoPdb

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  • MT1 receptor in Human [GtoPdb: 287] [UniProtKB: P48039]
  • This target only has 0 pki data point
1 _lig_chart_1 MT1 receptor Human
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  • MT2 receptor in Human [GtoPdb: 288] [UniProtKB: P49286]
  • This target only has 0 pki data point
2 _lig_chart_2 MT2 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MT1 receptor in Human [GtoPdb: 287] [UniProtKB: P48039]
GtoPdb - - 7.9 pEC50 12.59 nM EC50 Nature (2020) 579: 609-614 [PMID:32040955]
MT2 receptor in Human [GtoPdb: 288] [UniProtKB: P49286]
GtoPdb - - 6.2 pEC50 630.98 nM EC50 Nature (2020) 579: 609-614 [PMID:32040955]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.